Journal
ACS Medicinal Chemistry Letters
Published here
17 counted works of 17 linked
| Year | Title | Academics | Sources |
|---|---|---|---|
| 2021 | Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead. | William Jorgensen | CV OA |
| 2021 | Optimization of Triarylpyridinone Inhibitors of the Main Protease of SARS-CoV-2 to Low-Nanomolar Antiviral Potency. | William Jorgensen | CV OA |
| 2020 | Discovery of a cyclic choline analog that inhibits anaerobic choline metabolism by human gut bacteria. | Emily Balskus | CV OA |
| 2020 | Identification of 14 Known Drugs as Inhibitors of the Main Protease of SARS-CoV-2. | William Jorgensen | CV OA GS |
| 2020 | Structure-Guided Identification of DNMT3B Inhibitors. | William Jorgensen | CV OA |
| 2018 | Design, Synthesis and Biological Evaluation of Allosteric Effectors that Enhance CO Release from Carboxyhemoglobin | Jeffrey D. Winkler | CV OA GS |
| 2018 | Synthesis and Biological Evaluation of an Indazole-Based Selective Protein Arginine Deiminase 4 (PAD4) Inhibitor | Jon Ellman | CV OA |
| 2018 | Synthesis and Structure-Activity Relationship Study of Biliatresone, a Plant Isoflavonoid That Causes Biliary Atresia | Jeffrey D. Winkler | CV OA GS |
| 2017 | Adding a Hydrogen Bond May Not Help: Naphthyridinone vs. Quinoline Inhibitors of Macrophage Migration Inhibitory Factor. | William Jorgensen | CV OA |
| 2017 | Identification and Characterization of Small Molecules Binding to the JAK2 Pseudokinase Domain. | William Jorgensen | CV OA |
| 2017 | JAK2-JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules. | William Jorgensen | CV OA |
| 2017 | Systematic Study of Effects of Structural Modifications on the Aqueous Solubilities of Drug-like Molecules. | William Jorgensen | CV OA |
| 2016 | Cellular Activity of New Small Molecule Protein Arginine Deiminase 3 (PAD3) Inhibitors | Jon Ellman | CV OA |
| 2016 | Design, Conformation, and Crystallography of 2-Naphthyl Phenyl Ethers as Potent Anti-HIV Agents | William Jorgensen | CV OA |
| 2016 | Lee, W.-G.; Chan, A. H.; Spasov, K.A.; Anderson, K. A.; Jorgensen, W. L. | William Jorgensen | CV |
| 2015 | Potent Inhibitors Active Against HIV Reverse Transcriptase with K101P, a Mutation Conferring Rilpivirine Resistance | William Jorgensen | CV OA |
| 2014 | Picomolar Inhibitors of HIV-1 Reverse Transcriptase: Design and Crystallography of Naphthyl Phenyl Ethers | William Jorgensen | CV OA |