Trackademia

Welcome to Trackademia

The idea behind Trackademia is to build on existing academic databases like Google Scholar and OpenAlex so that you can trust the data and use it for whatever you want. That comes down to two things.

More data, and more ways to use it. We aggregate publication data from every major source into a single dataset and add information pulled from faculty CVs. Then we let you slice it however you want: choose which sources to build from, write your own formulas, weight journals, adjust for department size.

More accurate, and honest about where it isn’t. We focus on a smaller set of schools so we can verify everything carefully. Faculty lists come from department websites rather than being inferred from publication records, so we know who should be in the data before we go looking. When we can’t find data on someone, we record the gap instead of dropping them. Every number comes with a coverage rate you can check against ground truth.

Everything in Trackademia is built from seven units. AI merges duplicate records across sources and tags each publication so these categories hold up:

  • Publication — citation counts, authors, journal, peer review status, and more
  • Publication group — versions of the same work combined into one entity, such as a working paper and the article it became
  • Academic
  • Department
  • University
  • Field
  • Journal

There are two modes. In Database mode you browse the underlying records and filter by any of the seven units. In Analytics mode you get graphs and comparisons, and you switch views to compare two departments, compare one department against the average of the others, or see them all at once. Tabs let you focus on a particular level of the data.
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Academic

Jon Ellman

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Academic

RankDistinguished
As of2010 · CV
DepartmentYale Chemistry
UniversityYale
FieldChemistry
Scholarprofile

Totals

Publications356
Citations54,083
h-index123 · Scholar
Citations per year in post1,590.7
Years in post34 from the CV positions

Coverage

Works with a count345 of 356
Share97%

Positions

Eugene Higgins Professor of Chemistry, Yale U…2010–
Professor of Pharmacology, Yale University2010–
Professor of Cellular and Molecular Pharmacol…1999–2010
Professor of Chemistry, UC Berkeley1999–2010
Associate Professor of Chemistry, UC Berkeley1997–1998
Joel H. Hildebrand Associate Professor Chair…1996–1998
Assistant Professor of Chemistry, UC Berkeley1992–1997
National Science Foundation Postdoctoral Fell…1989–1992

Top venues 74 venues

The 8 holding the most of these works; 66 more hold at least one.

Journal of the American Chemical Society73
The Journal of Organic Chemistry49
Organic Letters43
Angewandte Chemie International Edition18
Bioorganic & Medicinal Chemistry Letters11
Journal of Medicinal Chemistry11
ChemInform7
Tetrahedron7

Publications per year

Works this academic published in each year, by the year each work appeared; an undated work is in no year, and a work two colleagues wrote counts for each of them. The kind, works and year filters decide which works are here at all.

Citations per year

Citations received in each year, from this academic’s verified Scholar profile, which counts every citation to everything they ever wrote: no publication filter reaches this line - not the kinds, not the works switch, not the year window on publication - and no journal weight either. It is a profile total, so it does not match the works listed below.

Publications 356 works

Every work these filters select, most cited first and the works with no count at the end: a work nobody has a figure for is unknown, never a zero to be ranked among the works that have one, and it prints an em dash. Each figure is that work’s own citations - Scholar’s count where there is one, else OpenAlex’s - and is not weighted.

YearTitleVenueKindCitations
2010Rhodium-Catalyzed C-C Bond Formation via Heteroatom-Directed C-H Bond ActivationChemical Reviewsarticle3,913
1996Synthesis and Applications of Small Molecule LibrariesChemical Reviewsarticle2,151
2012Rhodium Catalyzed Chelation-Assisted C–H Bond Functionalization ReactionsAccounts of Chemical Researcharticle1,491
2010Synthesis and Applications of tert-ButanesulfinamideChemical Reviewsarticle1,353
2002N-tert-Butanesulfinyl Imines: Versatile Intermediates for the Asymmetric Synthesis of AminesAccounts of Chemical Researcharticle1,093
2008Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed CH Bond ActivationAccounts of Chemical Researcharticle1,047
1997Catalytic Asymmetric Synthesis of tert-Butanesulfinamide. Application to the Asymmetric Synthesis of AminesJournal of the American Chemical Societyarticle788
1987Contrasteric Carboximide Hydrolysis with Lithium HydroperoxideTetrahedron Lettersarticle766
1992General and Expedient Method for the Solid-Phase Synthesis of 1,4-Benzodiazepine DerivativesJournal of the American Chemical Societyarticle756
2000Rapid and General Profiling of Protease Specificity by Using Combinatorial Fluorogenic Substrate LibrariesProceedings of the National Academy of Sciencesarticle740
2017Transition-Metal-Catalyzed C–H Bond Addition to Carbonyls, Imines, and Related Polarized π BondsChemical Reviewsarticle726
1999The Synthesis of Enantiomerically Pure N-tert-Butanesulfinyl Imines (tert-Butanesulfinimines) by the Direct Condensation of tert-Butanesulfinamide with Aldehyd…The Journal of Organic Chemistryarticle709
1990The Asymmetric Synthesis of -Amino Acids. Electrophilic Azidation of Chiral Imide Enolates, a Practical Approach to the Synthesis of (R)- and (S)--Azido Carb…Journal of the American Chemical Societyarticle693
2006Substrate Profiling of Cysteine Proteases Using a Combinatorial Peptide Library Identifies Functionally Unique SpecificitiesJournal of Biological Chemistryarticle561
1991A Biosynthetic Method for Introducing Unnatural Amino Acids Site-Specifically into ProteinsMethods in enzymology on CD-ROM/Methods in enzymologyarticle524
1999Asymmetric Synthesis of Chiral Amines by Highly Diastereoselective 1,2-Additions of Organometallic Reagents to N-tert-Butanesulfinyl IminesTetrahedronarticle491
2010Catalytic C-O Bond Cleavage of 2-Aryloxy-1-arylethanols and Its Application to the Depolymerization of Lignin Related PolymersJournal of the American Chemical Societyarticle490
1999Fmoc-BasedSynthesis of Peptide-Thioesters: Application to the Total Chemical Synthesis of a Glycoprotein by Native Chemical LigationJournal of the American Chemical Societyarticle484
1998ChemInform Abstract: Catalytic Asymmetric Oxidation of tert‐Butyl Disulfide. Synthesis of tert‐Butanesulfinamides, tert‐Butyl Sulfoxides, and tert‐Butanesulfin…ChemInformarticle479
1994The Combinatorial Synthesis, and Chemical and Biological Evaluation of a 1,4-Benzodiazepine LibraryProceedings of the National Academy of Sciencesarticle462
2015Cobalt(III)-Catalyzed Synthesis of Indazoles and Furans by C–H Bond Functionalization/Addition/Cyclization CascadesJournal of the American Chemical Societyarticle449
2008Synthesis of Dihydropyridines and Pyridines from Imines and Alkynes via C-H ActivationOSTI OAI (U.S. Department of Energy Office of Scientific an…article438
1992Site-Specific Incorporation of Novel Backbone Structures into ProteinsSciencearticle389
1996Design, Synthesis, and Evaluation of Small-Molecule LibrariesAccounts of Chemical Researcharticle386
2007Rh(I)-Catalyzed Alkylation of Quinolines and Pyridines via C-H Bond ActivationJournal of the American Chemical Societyarticle379
1998Catalytic Asymmetric Oxidation of tert-Butyl Disulfide. Synthesis of tert-Butanesulfinamides, tert-Butyl Sulfoxide, and tert-ButanesulfiniminesJournal of the American Chemical Societyarticle361
2000Synthesis of positional-scanning libraries of fluorogenic peptide substrates to define the extended substrate specificity of plasmin and thrombinNature Biotechnologyarticle355
2008Rh(I)-Catalyzed Direct Arylation of Pyridines and QuinolinesJournal of the American Chemical Societyarticle345
2002Peptide Microarrays for the Determination of Substrate SpecificityJournal of the American Chemical Societyarticle342
1999An Alkanesulfonamide “Safety-Catch” Linker for Solid-Phase SynthesisThe Journal of Organic Chemistryarticle338
1996Activation Method to Prepare a Highly Reactive Acylsulfonamide “Safety-Catch” Linker for Solid-Phase SynthesisJournal of the American Chemical Societyarticle336
2003Applications of tert-Butanesulfinamide in the Asymmetric Synthesis of AminesPure and Applied Chemistryarticle335
2013Rhodium(III)-Catalyzed Indazole Synthesis by C-H Bond Functionalization and Cyclative CaptureJournal of the American Chemical Societyarticle328
1991A General and Efficient Route for Chemical Aminoacylation of Transfer RNAsJournal of the American Chemical Societyarticle321
2011Rhodium(III)-Catalyzed Arylation of Boc-Imines via C-H Bond FunctionalizationJournal of the American Chemical Societyarticle316
1999The Asymmetric Synthesis of -Dibranched Amines by the Trimethylaluminum Mediated 1,2-Addition of Organolithiums to tert-Butanesulfinyl KetiminesJournal of the American Chemical Societyarticle308
2011Expedient Synthesis of N-Acyl Anthranilamides and β-Enamine Amides by the Rh(III)-Catalyzed Amidation of Aryl and Vinyl CH Bonds with IsocyanatesJournal of the American Chemical Societyarticle305
2000Combinatorial Target-Guided Ligand Assembly. Identification of Potent, Sub-type Selective c-Src InhibitorsProceedings of the National Academy of Sciencesarticle303
2011Rh(III)-Catalyzed Oxidative Coupling of Unactivated Alkenes via CH ActivationOrganic Lettersarticle302
2004Highly Efficient and Enantioselective Cyclization of Aromatic Imines via Directed C-H Bond ActivationJournal of the American Chemical Societyarticle302
1995Silicon-Based Linkage Strategy for Traceless Solid-Phase SynthesisThe Journal of Organic Chemistryarticle296
1999The tert-Butanesulfinyl Group: An Ideal Chiral Directing Group and Boc-Surrogate for Asymmetric -Amino Acid Synthesis and ApplicationsThe Journal of Organic Chemistryarticle294
2022Bespoke library docking for 5-HT2A receptor agonists with antidepressant activityNaturearticle286
2008Rh(I)-Catalyzed Arylation of Heterocycles via C-H Bond Activation: Expanded Scope Through Mechanistic Insight.Journal of the American Chemical Societyarticle285
2004Arylation of Heterocycles via Rhodium-Catalyzed C-H Bond FunctionalizationOrganic Lettersarticle284
1994Straightforward and General Method for Coupling Alcohols to Solid-SupportsTetrahedron Lettersarticle284
2008Asymmetric Copper-Catalyzed Synthesis of -Amino Boronate Esters from N-tert-Butanesulfinyl AldiminesJournal of the American Chemical Societyarticle277
1994Carbon-Carbon Bond Forming Methods on Solid Support. Utilization of Kenner's "Safety-Catch" LinkerJournal of the American Chemical Societyarticle275
1997Structure-Based Design and Combinatorial Chemistry Yield Low Nanomolar Inhibitors of Cathepsin DChemistry & Biologyarticle267
2001Annulation of Aromatic Imines via Directed C-H Activation with Wilkinson’s CatalystJournal of the American Chemical Societyarticle259
2005Total Synthesis of (+)-Lithospermic Acid by Asymmetric Intramolecular Alkylation via Catalytic C-H Bond ActivationJournal of the American Chemical Societyarticle251
1997The Solid-Phase Synthesis of 1,4-Benzodiazepine-2,5-diones. Library Preparation and Demonstration of Synthesis GeneralityThe Journal of Organic Chemistryarticle251
2007Enantioselective Aza-Henry Reaction with an N-Sulfinyl Urea OrganocatalystJournal of the American Chemical Societyarticle250
2002Intermediacy of an N-Heterocyclic Carbene in the Catalytic C-H Activation of BenzimidazoleJournal of the American Chemical Societyarticle243
2005Diastereoselective and Enantioselective Rh(I)-Catalyzed Additions of Arylboronic Acids to N-tert-Butanesulfinyl and N-Diphenylphosphinoyl AldiminesJournal of the American Chemical Societyarticle239
1999Single Digit Nanomolar, Low Molecular Weight Non-Peptide Inhibitors of Malarial Aspartyl Protease Plasmepsin IIJournal of Medicinal Chemistryarticle234
1995Combinatorial Asymmetric Catalyst Development. General Solid-Phase Synthesis Strategy for the Preparation of 2-Pyrrolidinemethanol LigandsThe Journal of Organic Chemistryarticle234
2003Catalytic Properties and Inhibition of Proline-Specific Dipeptidyl Peptidases II, IV and VIIBiochemical Journalarticle233
2002Asymmetric Synthesis of -Amino Acid Derivatives Incorporating a Broad Range of Substitution Patterns by Enolate Additions to tert-Butanesulfinyl IminesThe Journal of Organic Chemistryarticle233
1995Stille Coupling in the Solid Phase Synthesis of Structurally Diverse 1,4-Benzodiazepine DerivativesJournal of the American Chemical Societyarticle230
2013Facile Synthesis of Unsymmetrical Acridines and Phenazines by a Rhodium(III)-Catalyzed Amination, Cyclization and Aromatization CascadeJournal of the American Chemical Societyarticle227
2001Annulation of Alkenyl-Substituted Heterocycles via Rhodium-Catalyzed Intramolecular C-H Activated Coupling ReactionsJournal of the American Chemical Societyarticle226
2003Development and Application of a New General Method for the Asymmetric Synthesis of s yn - and a nti -1,3-Amino AlcoholsJournal of the American Chemical Societyarticle225
1989The Total Synthesis of the Isodityrosine-Derived Cyclic Tripeptides OF4949-III and K-13. Determination of the Absolute Configuration of K-13Journal of the American Chemical Societyarticle225
1995An expedient and high-yielding method for the solid-phase synthesis of diverse 1,4-benzodiazepine-2,5-dionesThe Journal of Organic Chemistryarticle222
2006Experimental and Computational Studies on the Mechanism of N-Heterocycle C-H Activation by Rh(I)Journal of the American Chemical Societyarticle220
1987Asymmetric Halogenation of Chiral Imide Enolates. A General Approach to the Synthesis of Enantiomerically Pure -Amino AcidsTetrahedron Lettersarticle219
2003An Improved Synthesis of tert-Butanesulfinamide Suitable for Large Scale ProductionOrganic Lettersarticle217
1995Expedient Method for the Solid-Phase Synthesis of Aspartic Acid Protease Inhibitors Directed toward the Generation of LibrariesJournal of Medicinal Chemistryarticle213
1994Simultaneous Solid-Phase Synthesis of -Turn Mimetics Incorporating Side-chain FunctionalityJournal of the American Chemical Societyarticle211
1992Probing Protein Stability with Unnatural Amino AcidsSciencearticle205
2002Expedient Solid-Phase Synthesis of Fluorogenic Protease Substrates Using the 7-Amino-4-Carbamoylmethylcoumarin (ACC) FluorophoreThe Journal of Organic Chemistryarticle201
2006NMR Shifts, Orbitals, and M···H-X Bonding in d8 Square Planar Metal ComplexesOrganometallicsarticle199
2001-Turn Mimetic Library Synthesis: Scaffolds and ApplicationsTetrahedronarticle195
1997Germanium and Silicon Linking Strategies for Traceless Solid-Phase SynthesisThe Journal of Organic Chemistryarticle193
2005High Throughput Substrate Specificity Profiling of Serine and Cysteine Proteases Using Solution-Phase Fluorogenic Peptide MicroaraysMolecular & Cellular Proteomicsarticle192
2010Rhenium-Catalyzed Didehydroxylation of Vicinal Diols to Alkenes Using a Simple Alcohol as a Reducing AgentJournal of the American Chemical Societyarticle190
2009Enantioselective Addition of Thioacetic Acid to Nitroalkenes via N-Sulfinyl Urea OrganocatalysisJournal of the American Chemical Societyarticle188
2003Novel Uncomplexed and Complexed Structures of Plasmepsin II, an Aspartic Protease from Plasmodium falciparumJournal of Molecular Biologyarticle187
2012Mechanism of the Rhodium(III)-Catalyzed Arylation of Imines via C–H Bond Functionalization: Inhibition by SubstrateJournal of the American Chemical Societyarticle185
2006The Total Synthesis of Tubulysin DJournal of the American Chemical Societyarticle185
2002Intermolecular Coupling of Alkenes to Heterocycles via Rhodium-Catalyzed C-H Bond ActivationJournal of the American Chemical Societyarticle183
2008Identification of a New Class of Nonpeptidic Inhibitors of CruzainJournal of the American Chemical Societyarticle180
2013Rhodium(III)-Catalyzed Alkenyl C-H Bond Functionalization: Convergent Synthesis of Furans and PyrrolesAngewandte Chemie International Editionarticle175
2002Asymmetric Synthesis of syn- and anti-1,3-Amino AlcoholsChemInformarticle175
2010Nonpeptidic Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors as Promising New Leads for Chagas Disease ChemotherapyJournal of Medicinal Chemistryarticle174
2006Enantioselective Synthesis of a PKC Inhibitor via Catalytic C-H Bond ActivationOrganic Lettersarticle174
2006Microwave-Promoted Rhodium-Catalyzed Arylation of Heterocycles through CH Bond ActivationAngewandte Chemie International Editionarticle172
1991Construction of a Caged Protein by Site-Specific Unnatural Amino Acid MutagenesisJournal of the American Chemical Societyarticle172
2001Asymmetric Synthesis of 1,2-Amino Alcohols Using tert-Butanesulfinyl Aldimines and KetiminesThe Journal of Organic Chemistryarticle170
2006Asymmetric Synthesis of Protected Arylglycines by Rhodium-Catalyzed Addition of Arylboronic Acids to N-tert-Butanesulfinyl Imino EstersJournal of the American Chemical Societyarticle166
2008Enantioselective Intramolecular Hydroarylation of Alkenes via Directed C-H Bond ActivationThe Journal of Organic Chemistryarticle165
2015Cobalt(III)-Catalyzed C–H Bond Amidation with IsocyanatesOrganic Lettersarticle162
2022Catalytic Enantioselective Sulfur Alkylation of Sulfenamides for the Asymmetric Synthesis of SulfoximinesJournal of the American Chemical Societyarticle161
2014Inhibitor of the Tyrosine Phosphatase STEP Reverses Cognitive Deficits in a Mouse Model of Alzheimer’s DiseasePLoS Biologyarticle161
2016Highly Stereoselective Cobalt(III)-Catalyzed Three-Component C−H Bond Addition CascadeAngewandte Chemie International Editionarticle160
2012Synthesis of Pyridines from Ketoximes and Terminal Alkynes via C–H Bond FunctionalizationThe Journal of Organic Chemistryarticle156
2003Microwave Assisted C-H Bond Activation: A Rapid Entry into Functionalized HeterocyclesOrganic Lettersarticle155
2005Profiling Serine Protease Substrate Specificity with Solution Phase Fluorogenic Peptide MicroarraysPROTEOMICSarticle147
2005Substrate Activity Screening: A Fragment-Based Method for the Rapid Identification of Nonpeptidic Protease InhibitorsJournal of the American Chemical Societyarticle146
1999One-pot asymmetric synthesis of tert-butanesulfinyl-protected amines from ketones by the in situ reduction of tert-butanesulfinyl ketiminesTetrahedron Lettersarticle146
2006Stereoselective Alkylation of α,-Unsaturated Imines via C-H Bond ActivationJournal of the American Chemical Societyarticle144
2004Catalytic Enantioselective Synthesis of Sulfinate Esters Through the Dynamic Resolution of tert-Butanesulfinyl ChlorideJournal of the American Chemical Societyarticle144
2001Synthesis, Utility, and Structure of Novel Bis(sulfinyl)imidoamidine Ligands for Asymmetric Lewis Acid CatalysisJournal of the American Chemical Societyarticle144
1999Combinatorial Library Approach to the Development of Synthetic Receptors Targeting Vancomycin Resistant BacteriaJournal of the American Chemical Societyarticle144
2003Crystal Structures of Reversible Ketone-Based Inhibitors of the Cysteine Protease CruzainBioorganic & Medicinal Chemistryarticle143
2012Highly Diastereoselective Synthesis of Tetrahydropyridines by a C–H Activation–Cyclization–Reduction CascadeJournal of the American Chemical Societyarticle141
1997A Silicon Linker for the Direct Loading of Aromatic Compounds onto Solid Supports. Traceless Synthesis of Pyridyl-Based TricyclicsThe Journal of Organic Chemistryarticle138
2003Enantioselective Oxidation of Di-tert-Butyl Disulfide with a Vanadium Catalyst: Progress toward Mechanism ElucidationThe Journal of Organic Chemistryarticle137
2017Rh(III)-Catalyzed Aryl and Alkenyl C–H Bond Addition to Diverse NitroalkenesACS Catalysisarticle136
2007One-Pot Asymmetric Synthesis of Either Diastereomer of tert-Butanesulfinyl-protected Amines from KetonesThe Journal of Organic Chemistryarticle136
2005Preagostic Rh-H Interactions and C-H Bond Functionalization: A Combined Experimental and Theoretical Investigation of Rhodium(I) Phosphinite ComplexesOrganometallicsarticle135
2007Fragment-Based Substrate Activity Screening method for the Identification of Potent Inhibitors of the M. tuberculosis Phosphatase PtpBJournal of the American Chemical Societyarticle133
2004Asymmetric -Alkylation of N'-tert-Butanesulfinyl Amidines. Application to the Total Synthesis of (6R,7S)-7-Amino-7,8-dihydro- -bisaboleneChemInformarticle131
1989The Oxidative Macrocyclization of Phenolic Peptides. A Biomimetic Approach to the Synthesis of the Vancomycin Family of AntibioticsJournal of the American Chemical Societyarticle131
2012A Nonpeptidic Cathepsin S Activity-Based Probe for Noninvasive Optical Imaging of Tumor-Associated MacrophagesChemistry & Biologyarticle130
2003Synthesis of a Tricyclic Mescaline Analog by Catalytic C-H Bond ActivationOrganic Lettersarticle129
2019α-Branched Amines by Catalytic 1,1-Addition of C–H Bonds and Aminating Agents to Terminal AlkenesNature Catalysisarticle124
2004Intermolecular Coupling of Alkenes to Heterocycles via C-H Bond ActivationThe Journal of Organic Chemistryarticle123
2010Aminopeptidase Fingerprints, an Integrated Approach for Identification of Good Substrates and Optimal InhibitorsJournal of Biological Chemistryarticle122
2008Asymmetric Synthesis of (−)-Incarvillateine Employing an Intramolecular Alkylation via Rh-Catalyzed Olefinic C−H Bond ActivationJournal of the American Chemical Societyarticle122
2002Benzodiazepine-Induced Superoxidce Signals B Cell Apoptosis: Mechanistic Insight and Potential Therapeutic UtilityJournal of Clinical Investigationarticle120
2009Recycling the tert-Butanesulfinyl Group in the Synthesis of Amines Using tert-ButanesulfinamideThe Journal of Organic Chemistryarticle118
1999Identification of a Potent Heterocyclic Ligand to Somatostatin Receptor Sub-Type 5 by the Synthesis and Screening of -Turn Mimetic LibrariesJournal of the American Chemical Societyarticle118
2009An Efficient Didehydroxylation Method for the Biomass-Derived Polyols Glycerol and Erythritol. Mechanistic Studies of a Formic Acid-Mediated DeoxygenationChemical Communicationsarticle117
2007Synthesis of Potent Bicyclic Bisarylimidazole c-Jun N-Terminal Kinase Inhibitors by Catalytic C-H Bond ActivationJournal of the American Chemical Societyarticle117
2002Combinatorial Strategies for Targeting Protein Families. Application to the ProteasesChemBioChemarticle117
2006Identification of Selective, Nonpeptidic Nitrile Inhibitors of Cathepsin S using the Substrate Activity Screening MethodJournal of Medicinal Chemistryarticle115
2003Novel Sulfinyl Imine Ligands for Asymmetric CatalysisOrganic Lettersarticle115
1993Protein Biosynthesis with Conformationally Restricted Amino AcidsJournal of the American Chemical Societyarticle114
2007Design, Synthesis, and Biological Properties of Highly Potent Tubulysin D AnaloguesChemistry - A European Journalarticle113
2005Annulation of Aromatic Imines via Directed C-H Bond ActivationThe Journal of Organic Chemistryarticle113
2018Rhodium(III)-Catalyzed Imidoyl C−H Activation for Annulations to AzolopyrimidinesOrganic Lettersarticle112
2009Asymmetric Synthesis of α–Branched Allylic Amines by the Rh(I)-Catalyzed Addition of Alkenyltrifluoroborates to N-tert-Butanesulfinyl AldiminesJournal of the American Chemical Societyarticle110
1998General Solid-Phase Synthesis Approach to Prepare Mechanism-Based Aspartyl Protease Inhibitor Libraries. Identification of Potent Cathepsin D InhibitorsJournal of the American Chemical Societyarticle110
1997Approaches to the Synthesis of the Vancomycin Antibiotics. Synthesis of Orienticin C (Bis-dechlorovancomycin) AglyconJournal of the American Chemical Societyarticle109
2012Rhodium-Catalyzed Synthesis of Branched Amines by Direct Addition of Benzamides to IminesOrganic Lettersarticle108
2001Design, Synthesis, and Utility of Support-Bound tert-ButanesulfinamideJournal of the American Chemical Societyarticle107
2012Rhodium(III)-Catalyzed Synthesis of Phthalides by Cascade Addition and Cyclization of Benzimidates with AldehydesChemical Sciencearticle105
2001Asymmetric Synthesis of Pre-Protected ,-Disubstituted Amino Acids from tert-Butanesulfinyl KetiminesTetrahedron Lettersarticle104
1997Solid Support Linker StrategiesChemInformarticle104
2010Rh(I)-Catalyzed Direct Arylation of AzinesThe Journal of Organic Chemistryarticle102
2003The Preparation and Utility of Bis(sulfinyl)imidoamidine Ligands for the Copper-Catalyzed Diels Alder ReactionThe Journal of Organic Chemistryarticle102
2000Novel Cathepsin D Inhibitors Block the Formation of Hyperphosphorylated Tau Fragments in HippocampusJournal of Neurochemistryarticle101
1996Expedient Synthesis of -Turn Mimetics Incorporating the i + 1, i + 2, and i + 3 SidechainsTetrahedron Lettersarticle101
2016Rh(III)-Catalyzed Diastereoselective C–H Bond Addition/Cyclization Cascade of Enone Tethered AldehydesChemical Sciencearticle100
1998Solid-Phase Synthesis of Diverse E- F-Series ProstaglandinsThe Journal of Organic Chemistryarticle100
2014Asymmetric Synthesis of α-Branched Amines via Rh(III)-Catalyzed C–H Bond FunctionalizationJournal of the American Chemical Societyarticle99
2012Catalytic Enantioselective Protonation of Nitronates Utilizing an Organocatalyst Chiral Only at SulfurJournal of the American Chemical Societyarticle99
2010Total Synthesis of (-)-AurantioclavineOrganic Lettersarticle99
2008Expedient Synthesis of N-Methyl Tubulysin Analogues with High CytotoxicityThe Journal of Organic Chemistryarticle98
2006Rhodium-Catalyzed Direct C-H Addition of 3,4-Dihydroquinazolines to Alkenes and Their Use in the Total Synthesis of VasicolineThe Journal of Organic Chemistryarticle97
2009Application of Daugulis Copper-Catalyzed Direct Arylation to the Synthesis of 5-Aryl BenzotriazepinesOrganic Lettersarticle96
2003Stereoselective Synthesis of 1,2-Disubstituted -Amino Alcohols by Nucleophilic Addition to N-tert-Butanesulfinyl aldiminesThe Journal of Organic Chemistryarticle96
2018Selective and Synergistic Cobalt(III)-Catalysed Three-Component C–H Bond Addition to Dienes and AldehydesNature Catalysisarticle95
2013Mechanistic Study of the Oxidative Coupling of Styrene with 2-Phenylpyridine Derivatives Catalyzed by Cationic Rhodium(III) via C–H ActivationJournal of the American Chemical Societyarticle95
1999Compounds that activate the mouse melanocortin-1 receptor identified by screening a small molecule library based upon the β-turnJournal of Medicinal Chemistryarticle95
1996Palladium-Mediated Three-Component Coupling Strategy for the Solid-Phase Synthesis of Tropane DerivativesThe Journal of Organic Chemistryarticle94
1999General Solid-phase Method for the Preparation of Mechanism-based Cysteine Protease InhibitorsJournal of the American Chemical Societyarticle93
2014Asymmetric Synthesis of Protected α-Amino Boronic Acid Derivatives with an Air- and Moisture-Stable Cu(II) CatalystThe Journal of Organic Chemistryarticle92
2002Identification of Potent and Selective Mechanism-Based Inhibitors of the Cysteine Protease Cruzain Using Solid-Phase Parallel SynthesisJournal of Medicinal Chemistryarticle92
2020Highly Diastereoselective Functionalization of Piperidines by Photoredox Catalyzed C–H Arylation and EpimerizationJournal of the American Chemical Societyarticle90
2011Highly Functional Group Compatible Rh-Catalyzed Addition of Arylboroxines to Activated N-tert-Butanesulfinyl KetiminesOrganic Lettersarticle90
2004Self-Condensation of N-tert-Butanesulfinyl Aldimines: Application to the Asymmetric Synthesis of Biologically Important Amine-Containing CompoundsOrganic Lettersarticle90
1997Combinatorial Thinking in Chemistry and BiologyProceedings of the National Academy of Sciencesarticle89
2014Convergent Synthesis of Diverse Tetrahydropyridines via Rh(I)-Catalyzed C–H Functionalization SequencesOrganic Process Research & Developmentarticle88
2001Definition of the Extended Substrate Specificity Determinants for -Tryptases I and IIJournal of Biological Chemistryarticle88
2015Design of a Highly Selective Quenched Activity-Based Probe and Its Application in Dual Color Imaging Studies of Cathepsin S Activity LocalizationJournal of the American Chemical Societyarticle86
2018Three-Component Coupling of Aldehydes, Aminopyrazoles, and Sulfoxonium Ylides via Rhodium(III)-Catalyzed Imidoyl C–H Activation: Synthesis of Pyrazolo[1,5-a]py…The Journal of Organic Chemistryarticle85
2002Altered Substrate Specificity of Drug-Resistant Human Immunodeficiency Virus Type 1 ProteaseJournal of Virologyarticle85
1992Site-Specific Isotopic Labeling of Proteins for NMR StudiesJournal of the American Chemical Societyarticle85
2021Rhodium-Catalyzed C–H Alkenylation/Electro-cyclization Cascade Provides Dihydropyridines That Serve as Versatile Intermediates to Diverse Nitrogen HeterocyclesAccounts of Chemical Researcharticle84
2013Proton Donor Acidity Controls Selectivity in Nonaromatic Nitrogen Heterocycle SynthesisSciencearticle84
2004Application of P,N-Sulfinyl Imine Ligands to Iridium-Catalyzed Asymmetric Hydrogenation of OlefinsThe Journal of Organic Chemistryarticle84
2008Positional-Scanning Fluorogenic Substrate Libraries Reveal Unexpected Specificity Determinants of Deubiquitinating Enzymes (DUBs)Biochemical Journalarticle83
2023Sulfur-Arylation of Sulfenamides via Chan–Lam Coupling with Boronic Acids: Access to High Oxidation State Sulfur PharmacophoresOrganic Lettersarticle82
2017A Convergent Synthesis of Functionalized Alkenyl Halides via Co(III)-Catalyzed Three-Component C-H Bond AdditionAngewandte Chemie International Editionarticle82
2010Functional studies of the Plasmodium falciparum dipeptidyl aminopeptidase I (DPAP1) using small molecule inhibitors and active siteChemistry & Biologyarticle82
2008Enantioselective Synthesis of -Aryl Alkylamines by Rh-Catalyzed Addition Reactions of Arylboronic Acids to Aliphatic IminesAngewandte Chemie International Editionarticle82
1999Chiral N-Acyl-tert-Butanesulfinamides: The “Safety-Catch” Principle Applied to Diastereoselective Enolate AlkylationsThe Journal of Organic Chemistryarticle81
2005A Rapid and General Method for the Asymmetric Synthesis of 2-Substituted Pyrrolidines Using tert-ButanesulfinamideOrganic & Biomolecular Chemistryarticle80
2001A Mass Spectrometric Labeling Strategy for High-Throughput Reaction Evaluation and Optimization: Exploring C–H ActivationPubMedarticle80
2007Catalytic Enantioselective Addition of Arylboronic Acids to N-Boc Imines Generated in SituOrganic Lettersarticle79
1999Synthesis of Alkoxylamines by Alkoxide Amination with 3,3‘-Di- tert -butyloxaziridineThe Journal of Organic Chemistryarticle77
2006Reassignment of Configuration for Salvianolic Acid B and Establishment of Its Identity with Lithospermic Acid BJournal of Natural Productsarticle76
2010Asymmetric Rh(I)-Catalyzed Addition of MIDA Boronates to N-tert-Butanesulfinyl Aldimines: Development and Comparison to TrifluoroboratesThe Journal of Organic Chemistryarticle75
2004Rhodium-Catalyzed Direct C-H Addition of 4,4-Dimethyl-2-oxazoline to AlkenesOrganic Lettersarticle75
1998Novel Inhibitors of 41 Integrin Receptor Interactions Through Library Synthesis and ScreeningBioorganic & Medicinal Chemistry Lettersarticle75
2003(RS)‐(+)‐2‐Methyl‐2‐propanesulfinamide [tert‐Butanesulfinamide]Organic Synthesesarticle74
1999Parallel Solid-Phase Synthesis of Prostaglandin E AnalogsJournal of Combinatorial Chemistryarticle74
2016Conjugate Addition–Enantioselective Protonation ReactionsBeilstein Journal of Organic Chemistryarticle73
2014Regio- and Stereoselective 1,2-Dihydropyridine Alkylation/Addition Sequence for the Synthesis of Piperidines with Quaternary CentersAngewandte Chemie International Editionarticle73
2015An Efficient Method for the Preparation of Styrene Derivatives via Rh(III)-Catalyzed Direct C–H VinylationOrganic Lettersarticle72
2017Synthesis of [5,6]-Bicyclic Heterocycles with a Ring-Junction Nitrogen via Rh(III)-Catalyzed C-H Functionalization of Alkenyl AzolesAngewandte Chemie International Editionarticle71
2012Enantio- and Diastereoselective Addition of Cyclohexyl Meldrum’s Acid to β- and α,β-Disubstituted Nitroalkenes via N-Sulfinyl Urea CatalysisChemInformarticle71
2010Identification and Evaluation of Novel Small Molecule Pan-Caspase Inhibitors in Huntington’s Disease ModelsChemistry & Biologyarticle71
2024Enantioselective S-Alkylation of Sulfenamides by Phase-Transfer CatalysisAngewandte Chemie International Editionarticle69
2023Preparation of Sulfilimines by Sulfur-Alkylation of N-Acyl Sulfenamides with Alkyl HalidesThe Journal of Organic Chemistryarticle68
2006Asymmetric Synthesis of ,-Dibranched Propargylamines by Acetylide Additions to N-tert-Butanesulfinyl KetiminesThe Journal of Organic Chemistryarticle68
2005Catalytic Enantioselective Sulfinyl Transfer Using Cinchona Alkaloid CatalystsOrganic Lettersarticle68
2012Conformational Change in Rhomboid Protease GlpG Induced by Inhibitor Binding to Its S′ SubsitesBiochemistryarticle67
2009Fragment-based discovery of selective inhibitors of the Mycobacterium tuberculosis protein tyrosine phosphatase PtpABioorganic & Medicinal Chemistry Lettersarticle67
2020Co(III)-Catalyzed C-H Amidation of Dehydroalanine for the Site-Selective Structural Diversification of ThiostreptonAngewandte Chemie International Editionarticle66
2017Base-Controlled Completely Selective Linear or Branched Rhodium(I)-Catalyzed C−H ortho-Alkylation of Azines without PreactivationAngewandte Chemie International Editionarticle66
2003Attenuation of Autoimmune Disease in Fas-Deficient Mice by Treatment with a Cytotoxic Benzodiazepine—article66
2003Parallel Solution-Phase Asymmetric Synthesis of -Branched AminesJournal of Combinatorial Chemistryarticle66
2005N-Sulfinyl Metalloenamine Conjugate Additions: Asymmetric Synthesis of PiperidinesThe Journal of Organic Chemistryarticle65
1995Photochemically-Initiated Protein SplicingAngewandte Chemie International Edition in Englisharticle65
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2013Unstabilized Azomethine Ylides for the Stereoselective synthesis of Substituted Piperidines, Tropanes and Azabicyclo[3.1.0] systemsJournal of the American Chemical Societyarticle61
2005Asymmetric Conjugate Addition of Copper Reagents to ,-Unsaturated tert-Butanesulfinyl IminesOrganic Lettersarticle61
1997Synthesis and Evaluation of a Library of Peptidomimetics Based upon the -TurnTetrahedronarticle60
2013Asymmetric Synthesis of Amines Using tert-ButanesulfinamideNature Protocolsarticle59
2010Synthesis of Multicyclic Pyridine and Quinoline Derivatives via Intramolecular C-H Bond FunctionalizationOrganic Lettersarticle59
2004Highly Stereoselective Addition of Organometallic Reagents to N- tert-Butanesulfinyl Imines Derived from 3- and 4-Substituted CyclohexanonesOrganic Lettersarticle59
2014Catalytic Enantioselective Addition of Thioacids to Trisubstituted NitroalkenesAngewandte Chemie International Editionarticle58
2002Tyrosylprotein Sulfotransferase Inhibitors Generated by Combinatorial Target-Guided ligand AssemblyBioorganic & Medicinal Chemistry Lettersarticle58
2013Synthesis of Isoquinuclidines from Highly Substituted Dihydropyridines via the Diels-Alder ReactionOrganic Lettersarticle57
1996Non-Nucleic Acid Inhibitors of Protein-DNA Interactions Identified through Combinatorial ChemistryJournal of the American Chemical Societyarticle57
2021Three-Component 1,2-Carboamidation of Bridged Bicyclic Alkenes via RhIII-Catalyzed Addition of C–H Bonds and Amidating ReagentsOrganic Lettersarticle54
2003D-Ala-D-Lac Binding is Not Required for the High Activity of Vancomycin Dimers Against Vancomycin Resistant EnterococciJournal of the American Chemical Societyarticle54
2019Synthesis of Homoallylic Alcohols with Acyclic Quaternary Centers via CoIII‐Catalyzed Three‐Component C–H Bond Addition to Internally Substituted Dienes and Ca…Angewandte Chemie International Editionarticle53
2011Development of an N-Sulfinyl Prolinamide for the Asymmetric Aldol ReactionTetrahedronarticle53
2003The Proapoptotic Benzodiazepine BZ-423 Affects the Growth and Survival of Malignant B CellsPubMedarticle53
2008Synthesis of a Benzodiazepine-derived Rhodium NHC Complex by C-H Bond ActivationOrganometallicsarticle52
2018Inhibition of STEP61 ameliorates deficits in mouse and hiPSC-based schizophrenia modelsMolecular Psychiatryarticle51
2011A Facile, Metal- and Solvent Free, Autoxidative Coupling of Quinolines with Indoles and PyrrolesChemical Communicationsarticle51
1998Synthesis of 3-Substituted 1,4-Benzodiazepin-2-onesJournal of the Brazilian Chemical Societyarticle51
2025Sulfilimines from a Medicinal Chemist’s Perspective: Physicochemical and in Vitro Parameters Relevant for Drug DiscoveryJournal of Medicinal Chemistryarticle49
2010Time-Resolved Single-Step Protease Activity Quantification Using Nanoplasmonic Resonator SensorsACS Nanoarticle49
2009Rhodium Catalyzed Enantioselective Cylization of Substituted Imidazoles via C–H Bond ActivationChemical Communicationsarticle49
2008The Stereoselective Formation of Bicyclic Enamines with Bridgehead Unsaturation via Tandem C-H Bond Activation/Alkenylation/ElectrocyclizationJournal of the American Chemical Societyarticle49
2021General Light-Mediated, Highly Diastereoselective Piperidine Epimerization: From Most Accessible to Most Stable StereoisomerJournal of the American Chemical Societyarticle48
2007Substrate Activity Acreening (SAS): a General Procedure for the Preparation and Screening of a Fragment-based Non-peptidic Protease Substrate Library for Inhib…Nature Protocolsarticle47
2021Pharmacological Inhibition of PI5P4Kα/β Disrupts Cell Energy Metabolism and Selectively Kills p53-Null Tumor CellsProceedings of the National Academy of Sciencesarticle46
2012Enantio- and Diastereoselective Addition of Thioacetic Acid to Nitroalkenes via N-Sulfinyl Urea CatalysisTetrahedronarticle45
2022C–H Bond Activation and Sequential Addition to Two Different Coupling Partners: A Versatile Approach to Molecular ComplexityChemical Society Reviewsarticle44
2018Rhodium(III)-Catalyzed C–H Functionalization of C-Alkenyl Azoles with Sulfoxonium Ylides for the Synthesis of Bridgehead N-Fused [5,6]-bicyclic HeterocyclesTetrahedronarticle44
2016Convergent Synthesis of Diverse Nitrogen Heterocycles via Rh(III)-Catalyzed C–H Conjugate Addition/Cyclization ReactionsOrganic Lettersarticle44
2013Substrate-Based Fragment Identification for the Development of Selective, Nonpeptidic Inhibitors of Striatal-Enriched Protein Tyrosine PhophataseJournal of Medicinal Chemistryarticle44
2011Chemotherapeutic Evaluation of a Novel Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing MiceChemMedChemarticle44
2015Synthesis of ent-Ketorfanol via a C–H Alkenylation/ Torquoselective 6π-Electrocyclization CascadeAngewandte Chemie International Editionarticle43
2011Asymmetric Synthesis of Amines by the Knochel-Type MgCl2-Enhanced Addition of Benzyl Zinc Reagents to N-tert-Butanesulfinyl AldiminesOrganic Lettersarticle43
2019Three-Component Coupling of Aldehydes, 2-Aminopyridines, and Diazo Esters via Rhodium(III)-Catalyzed Imidoyl C–H Activation: Synthesis of Pyrido[1,2-a]pyrimidi…Organic Lettersarticle42
2018Synthesis of Azolo[1,3,5]triazines via Rhodium(III)-Catalyzed Annulation of N-Azolo Imines and DioxazolonesThe Journal of Organic Chemistryarticle42
2003Structure Activity Studies of a Novel Cytotoxic BenzodiazepineBioorganic & Medicinal Chemistry Lettersarticle42
2015Facile Rh(III)-Catalyzed Synthesis of Fluorinated PyridinesOrganic Lettersarticle41
2014Convergent, Asymmetric Synthesis of Vicinal Amino Alcohols via Rh-Catalyzed Addition of α-Amido Trifluoroborates to CarbonylsChemical Sciencearticle41
2007Peptide-Nanocrescent Hybrid SERS Probe for Optical Detection of Protease ActivityJournal of Nanoscience and Nanotechnologyarticle41
2007Nonpeptidic Inhibitors of Cathepsin S with an Unprecedented Binding ModeJournal of Medicinal Chemistryarticle41
2025Ruthenium-Catalyzed Enantioselective Alkylation of Sulfenamides: A General Approach for the Synthesis of Drug Relevant S-Methyl and S-Cyclopropyl SulfoximinesJournal of the American Chemical Societyarticle40
2017Total Synthesis of (+)-Pancratistatin by the Rh(III)-Catalyzed Addition of a Densely Functionalized Benzamide to a Sugar-Derived NitroalkeneOrganic Lettersarticle40
2003Synthesis of a Diverse Library of Mechanism-Based Cysteine Protease InhibitorsJournal of Combinatorial Chemistryarticle40
2002Design and Synthesis of Novel Inhibitors of Gelatinase BBioorganic & Medicinal Chemistry Lettersarticle40
2015Identification of Multiple Structurally-Distinct, Nonpeptidic Small Molecule Inhibitors of Protein Arginine Deiminase 3 Using a Substrate-Based Fragment MethodJournal of the American Chemical Societyarticle39
2010ChemInform Abstract: Racemization Free Protocol for the Synthesis of N‐tert‐Butanesulfinyl Ketimines.ChemInformarticle38
2002Novel and Potent Anti-Malarial AgentsBioorganic & Medicinal Chemistryarticle38
2001Parallel Solution-Phase Synthesis of Mechanism-Based Cysteine Protease InhibitorsOrganic Lettersarticle37
1997The Synthesis of a 1680 Compound 1,4-Benzodiazepine LibraryNew Journal of Chemistryarticle37
2016Catalytic Enantioselective Addition of Pyrazol-5-ones to Trisubstituted Nitroalkenes with an N-Sulfinylurea OrganocatalystAdvanced Synthesis & Catalysisarticle36
2016Inhibition of the Tyrosine Phosphatase STEP61 Restores BDNF Expression and Reverses Motor and Cognitive Deficits in Phencyclidine-Treated MiceCellular and Molecular Life Sciencesarticle36
2016Preparation of Enantiomerically Pure Perfluorobutanesulfinamide and Its Application to the Asymmetric Synthesis of α-Amino AcidsThe Journal of Organic Chemistryarticle36
2017C2-Selective Branched Alkylation of Benzimidazoles by Rhodium(I)-Catalyzed C–H ActivationThe Journal of Organic Chemistryarticle35
2010Design and Synthesis of Novel Inhibitors for the Mycobacterium tuberculosis Phosphatase PtpBOrganic & Biomolecular Chemistryarticle35
2006Functional Phenotyping of Human Plasma Using a 361-Fluorogenic Substrate Biosensing MicroarrayBiotechnology and Bioengineeringarticle35
2003Identification of Potent and Broad-Spectrum Antibiotics from SAR Studies of a Synthetic Vancomycin AnalogBioorganic & Medicinal Chemistry Lettersarticle35
2016New Regio- and Stereoselective Cascades via Unstabilized Azomethine Ylide Cycloadditions for the Synthesis of Highly Substituted Tropane and Indolizidine Frame…Journal of the American Chemical Societyarticle34
2007Asymmetric Intramolecular Alkylation of Chiral Aromatic Imines via Catalytic C-H Bond ActivationSynlettarticle34
1996Synthesis and Evaluation of 1,4-Benzodiazepine LibrariesMethods in enzymology on CD-ROM/Methods in enzymologyarticle34
2017X-Ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase InhibitorsJournal of Medicinal Chemistryarticle33
2011A Fragmenting Hybrid Approach for Targeted Delivery of Multiple Therapeutic Agents to the Malaria ParasiteChemMedChemarticle33
2002Interference with Heme Binding to Histidine-Rich Protein-2 As an Antimalarial StrategyChemistry & Biologyarticle33
1999Benzodiazepine Compounds as Inhibitors of the Src Protein Tyrosine Kinase: Screening of a Combinatorial Library of 1,4-BenzodiazepinesArchives of Biochemistry and Biophysicsarticle33
2021Synthesis of Nitrile Bearing Acyclic Quaternary Centers via Co(III)‐Catalyzed Sequential C–H Bond Addition to Dienes and N‐CyanosuccinimideAngewandte Chemie International Editionarticle32
2000Asymmetric Synthesis of a C-3 Substituted Pipecolic AcidThe Journal of Organic Chemistryarticle32
2015Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors with Improved Pharmacokinetic Properties as Therapeutic Leads for Chagas’ DiseaseBioorganic & Medicinal Chemistry Lettersarticle30
2011Tubulysin D Analogues—article30
2018Rh(III)-Catalyzed Synthesis of Isoquinolones and 2-Pyridones via Annulation of N-Methoxyamides and NitroalkenesEuropean Journal of Organic Chemistryarticle29
2010Racemization Free Protocol for the Synthesis “N-tert-Butanesulfinyl KetimimesThe Journal of Organic Chemistryarticle29
2006Rapid Identification of Potent Nonpeptidic Serine Protease InhibitorsChemBioChemarticle29
2024Rh(II)-Catalyzed Enantioselective S-Alkylation of Sulfenamides with Acceptor–Acceptor Diazo Compounds Enables the Synthesis of Sulfoximines Displaying Diverse…Organic Lettersarticle28
2020Annulation of Hydrazones and Alkynes via Rhodium(III)-Catalyzed Dual C–H Activation: Synthesis of Pyrrolopyridazines and AzolopyridazinesOrganic Lettersarticle28
2016Rh(III)-Catalyzed C–H Bond Addition/Amine-Mediated Cyclization of Bis-Michael AcceptorsOrganic Lettersarticle28
2024Synthesis of N-Acylsulfenamides from (Hetero)Aryl Iodides and Boronic Acids by One-Pot Sulfur-Arylation and DealkylationAngewandte Chemie International Editionarticle27
2016Down-Regulation of BDNF in Cell and Animal Models Increases Striatal-Enriched Protein Tyrosine Phosphatase STEP61 LevelsJournal of Neurochemistryarticle27
2015Regio- and Diastereoselective Synthesis of Highly Substituted, Oxygenated Piperidines from TetrahydropyridinesThe Journal of Organic Chemistryarticle27
2014A Lewis Acid-Catalyzed Annulation to 2,1-BenzisoxazolesThe Journal of Organic Chemistryarticle27
2007The Direct ApproachSciencearticle27
1999Preparation of Enantioenriched α-Bromo Acids Incorporating Diverse FunctionalitySynthesisarticle27
—Anthony-Cahill, S., Noren, CJ, & Schultz, PG (1991)Methods in enzymology on CD-ROM/Methods in enzymologyarticle27
2023Synthesis of N-Acylsulfenamides from Amides and N-ThiosuccinimidesSynthesisarticle24
2022Stereoselective Synthesis of Allenyl Alcohols by Cobalt(III)-Catalyzed Sequential C−H Bond Addition to 1,3-Enynes and AldehydesAngewandte Chemie International Editionarticle24
2019Asymmetric Synthesis of (−)-NaltrexoneChemical Sciencearticle24
2020An allosteric site on MKP5 reveals a strategy for small molecule inhibitionScience Signalingarticle22
2017Glutathione-Responsive Selenosulfide Prodrugs as a Platform Strategy for Potent and Selective Mechanism-Based Inhibition of Protein Tyrosine PhosphatasesACS Central Sciencearticle22
2023Stereospecific Synthesis of Unprotected, α,β-Disubstituted Tryptamines and Phenethylamines from 1,2-Disubstituted Alkenes via a One-Pot Reaction SequenceOrganic Lettersarticle21
2022Visible Light-Mediated, Highly Diastereoselective Epimerization of Lactams from the Most Accessible to the More Stable StereoisomerACS Catalysisarticle21
2021Synthesis of α-Branched Amines by Three- and Four-Component C–H Functionalization Employing a Readily Diversifiable Hydrazone Directing GroupOrganic Lettersarticle21
2019The Breadth and Depth of C–H FunctionalizationThe Journal of Organic Chemistryarticle21

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